SCHEMBL6204424

SCHEMBL6204424

COc1ccc(C(C#N)CC(=O)c2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.69
KMT2A Q03164 2/20 0.67
NPC1 O15118 5/20 0.59
RAB9A P51151 5/20 0.59
ALDH1A1 P00352 4/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
TDP1 Q9NUW8 1/20 0.59
MAPT P10636 2/20 0.54
LMNA P02545 2/20 0.54
MGAM O43451 1/20 0.53
GAA P10253 1/20 0.53
SI P14410 1/20 0.53
MGAM2 Q2M2H8 1/20 0.53
FFAR1 O14842 1/20 0.50
NPSR1 Q6W5P4 2/20 0.49
PAX8 Q06710 1/20 0.49
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
POLB P06746 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8698087 0.94 L3MBTL1 (0.61) L3MBTL1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28727176 0.87 KMT2A (0.58) L3MBTL1KMT2ANPC1RAB9AALDH1A1
SCHEMBL13100658 0.86 KMT2A (0.79) L3MBTL1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL31326036 0.85 KMT2A (0.70) L3MBTL1KMT2ANPC1RAB9ACES2
SCHEMBL31326025 0.85 TSHR (0.53) L3MBTL1KMT2ANPC1ALDH1A1SMN1; SMN2
SCHEMBL1754734 0.85 TSHR (0.53) L3MBTL1KMT2ANPC1ALDH1A1SMN1; SMN2
SCHEMBL8695606 0.84 KMT2A (0.55) L3MBTL1KMT2ANPC1RAB9AALDH1A1
SCHEMBL25525563 0.84 KMT2A (0.55) L3MBTL1KMT2ANPC1RAB9AALDH1A1
SCHEMBL8697129 0.84 KMT2A (0.53) L3MBTL1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28727138 0.84 KMT2A (0.53) L3MBTL1KMT2ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015524-A1 IMPROVED PROCESS FOR THE SYNTHESIS OF BETA-KETONITRILES WARNER-LAMBERT COMPANY (US) 1998-04-16 WO claimed
CN-119504491-A Efficient preparation method and application of optically pure beta-cyano ketone 哈尔滨理工大学 2025-02-25 CN disclosed
CN-114456086-B Synthesis method of beta-cyano ketone 哈尔滨理工大学 2024-10-01 CN disclosed
CN-114456086-A Synthesis method of beta-cyano ketone 哈尔滨理工大学 2022-05-10 CN disclosed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
WO-1998015524-A1 IMPROVED PROCESS FOR THE SYNTHESIS OF BETA-KETONITRILES WARNER-LAMBERT COMPANY (US) 1998-04-16 WO disclosed
US-5416118-A Enzyme inhibitors SCHERING CORPORATION (US) 1995-05-16 US disclosed
EP-0583346-A1 BICYCLIC AMIDES AS INHIBITORS OF ACYL-COENZYME A: CHOLESTEROL ACYL TRANSFERASE SCHERING CORPORATION (US) 1994-02-23 EP disclosed
WO-1992018462-A1 BICYCLIC AMIDES AS INHIBITORS OF ACYL-COENZYME A: CHOLESTEROL ACYL TRANSFERASE SCHERING CORPORATION (US) 1992-10-29 WO disclosed
EP-0508425-A1 Bicyclic amides as inhibitors of acyl-coenzyme a: cholesterol acyl transferase SCHERING CORPORATION (US) 1992-10-14 EP disclosed