SCHEMBL6204532

SCHEMBL6204532

COc1ccc(C(=O)Cc2ccccc2)cc1C

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.56
TAS1R1 Q7RTX1 2/20 0.56
NPC1 O15118 3/20 0.53
HPGD P15428 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
MAPT P10636 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TAS2R14 Q9NYV8 1/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
GRM1 Q13255 1/20 0.48
PLAU P00749 1/20 0.48
KDM4E B2RXH2 1/20 0.48
SRD5A2 P31213 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257535 0.88 NPC1 (0.53) NPC1HPGDRAB9ASMN1; SMN2LMNA
SCHEMBL1515747 0.88 NPC1 (0.63) NPC1HPGDRAB9ASMN1; SMN2LMNA
SCHEMBL6575456 0.85 GAA (0.56) NPC1HPGDRAB9ASMN1; SMN2LMNA
SCHEMBL1515704 0.84 HTT (0.62) TAS1R3TAS1R1NPC1HPGDRAB9A
SCHEMBL29236861 0.84 LMNA (0.54) TAS1R3TAS1R1NPC1SMN1; SMN2LMNA
SCHEMBL7220907 0.84 MAPT (0.55) TAS1R3TAS1R1NPC1HPGDRAB9A
SCHEMBL14982198 0.83 NPC1 (0.60) TAS1R3TAS1R1NPC1HPGDRAB9A
SCHEMBL7040136 0.82 CES2 (0.58) NPC1RAB9ASMN1; SMN2LMNAMAPT
SCHEMBL6060544 0.82 HTT (0.61) NPC1HPGDRAB9ASMN1; SMN2HTT
SCHEMBL7047105 0.81 SMN1; SMN2 (0.80) NPC1HPGDRAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed