SCHEMBL6204872

SCHEMBL6204872

CCOc1cccc2c(=O)c(C(=O)NCc3ccc(Cn4ccnc4)cc3)c[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NPC1 O15118 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
RAB9A P51151 1/20 0.47
MAPK10 P53779 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ELANE P08246 1/20 0.45
ADORA2A P29274 5/20 0.45
WDR5 P61964 2/20 0.44
FLT3 P36888 1/20 0.42
TYRO3 Q06418 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207242 0.86 ADORA2A (0.47) ELANEADORA2AWDR5ADORA1
SCHEMBL6205058 0.82 POLB (0.62) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6204974 0.82 POLB (0.64) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6206617 0.82 POLB (0.50) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6204863 0.82 POLB (0.68) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6203895 0.81 POLB (0.49) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6206261 0.81 ADORA2A (0.55) POLBALDH1A1MEN1KMT2ANPC1
SCHEMBL6205541 0.81 MEN1 (0.52) POLBMEN1KMT2ANPC1RAB9A
SCHEMBL6206694 0.80 WDR5 (0.47) POLBRAB9AELANEADORA2AWDR5
SCHEMBL6205372 0.79 POLB (0.55) POLBALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed