SCHEMBL6206261

SCHEMBL6206261

CCOc1cccc2c(=O)c(C(=O)NCc3cccnc3)c[nH]c12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.55
LMNA P02545 3/20 0.55
HPGD P15428 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
KDM4E B2RXH2 2/20 0.55
TP53 P04637 1/20 0.55
HTT P42858 1/20 0.55
MAPK1 P28482 2/20 0.53
ALDH1A1 P00352 5/20 0.52
POLB P06746 3/20 0.52
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 3/20 0.52
RAB9A P51151 2/20 0.52
CYP2C19 P33261 2/20 0.52
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
MAPK10 P53779 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204974 0.88 POLB (0.64) ADORA2AHPGDSMN1; SMN2KDM4ETP53
SCHEMBL6205058 0.84 POLB (0.62) ADORA2ALMNAHPGDSMN1; SMN2KDM4E
SCHEMBL6206717 0.83 POLB (0.54) ADORA2AHPGDSMN1; SMN2TP53ALDH1A1
SCHEMBL6204593 0.83 ALDH1A1 (0.56) ADORA2ALMNAHPGDSMN1; SMN2KDM4E
SCHEMBL6205974 0.82 POLB (0.57) ADORA2AHPGDSMN1; SMN2TP53ALDH1A1
SCHEMBL6207376 0.81 POLB (0.58) ADORA2AHPGDSMN1; SMN2KDM4ETP53
SCHEMBL6204872 0.81 POLB (0.47) ADORA2AHPGDSMN1; SMN2TP53ALDH1A1
SCHEMBL6206629 0.81 POLB (0.56) ADORA2AHPGDSMN1; SMN2TP53ALDH1A1
SCHEMBL6206084 0.81 POLB (0.79) ADORA2ALMNAHPGDSMN1; SMN2KDM4E
SCHEMBL6205372 0.80 POLB (0.55) ADORA2ALMNAHPGDSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed