SCHEMBL6205063

SCHEMBL6205063

CC(C)c1nnc(NC(=O)Nc2ccc(F)c(COc3cccnc3)c2)s1.Nc1ccc(F)c(COc2cccnc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 4/20 0.46
MAPT P10636 4/20 0.46
GLA P06280 2/20 0.46
TSHR P16473 2/20 0.46
LMNA P02545 2/20 0.46
MAPK14 Q16539 1/20 0.43
BLM P54132 3/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
MAPK1 P28482 1/20 0.39
G6PD P11413 1/20 0.39
USP2 O75604 1/20 0.38
PKM P14618 1/20 0.38
PTPRE P23469 1/20 0.38
HTT P42858 2/20 0.38
TP53 P04637 1/20 0.38
HPN P05981 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080170 0.95 NPC1 (0.51) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6309454 0.87 NPC1 (0.43) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6079674 0.82 RAB9A (0.49) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6206155 0.77 MAPK14 (0.49) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL6080069 0.74 NOS1 (0.47) RAB9AMAPTLMNA
SCHEMBL6309458 0.74 NPC1 (0.40) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6204115 0.72 PTPRE (0.41) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6226761 0.72 MAPK14 (0.61) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL6079321 0.72 MAPK14 (0.54) MEN1KMT2AMAPTLMNAMAPK14
SCHEMBL6078757 0.71 RAB9A (0.56) NPC1RAB9AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545523-A1 3-&-grave;(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES ASP38 MAP KINASE INHIBITORS Astex Technology Limited (GB) 2005-06-29 EP disclosed
WO-2004004720-A1 3-`(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES AS P38 MAP KINASE INHIBITORS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO disclosed