SCHEMBL6309458

SCHEMBL6309458

CC(C)c1nnc(NC(=O)N(c2ccc(F)c(COc3cccnc3)c2)N(F)c2cccc(COc3cccnc3)c2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.40
RAB9A P51151 8/20 0.40
ALDH1A1 P00352 6/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
G6PD P11413 1/20 0.37
MAPK1 P28482 1/20 0.35
GPR132 Q9UNW8 3/20 0.35
GRM2 Q14416 1/20 0.35
NOX1 Q9Y5S8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.33
USP2 O75604 1/20 0.33
PKM P14618 1/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6309454 0.78 NPC1 (0.43) NPC1RAB9AALDH1A1SMN1; SMN2G6PD
SCHEMBL6080170 0.78 NPC1 (0.51) NPC1RAB9AALDH1A1SMN1; SMN2G6PD
SCHEMBL6205063 0.74 NPC1 (0.46) NPC1RAB9AALDH1A1SMN1; SMN2G6PD
SCHEMBL6079674 0.66 RAB9A (0.49) NPC1RAB9AALDH1A1SMN1; SMN2MAPK1
SCHEMBL6206155 0.63 MAPK14 (0.49) NPC1RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL6230436 0.62 SIRT2 (0.57) RAB9ASIRT2SIRT1SIRT3
SCHEMBL19702030 0.61 NOS1 (0.50) NPC1RAB9ASMN1; SMN2MAPK1GPR132
SCHEMBL6080064 0.60 MAOB (0.53) SMN1; SMN2KMT2ASIRT2SIRT1SIRT3
SCHEMBL6078757 0.60 RAB9A (0.56) NPC1RAB9AALDH1A1SMN1; SMN2MEN1
SCHEMBL6078971 0.60 MAPK14 (0.56) MAPK1SIRT2SIRT1SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002673-A1 RAF KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed