SCHEMBL6205783

SCHEMBL6205783

CN(C)/C=C/C(=O)c1c(-c2cccc(C(F)(F)F)c2)nn2ncccc12

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
GSK3B P49841 8/20 0.44
GAA P10253 1/20 0.42
TDP1 Q9NUW8 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
TRPV1 Q8NER1 2/20 0.39
KCNH2 Q12809 1/20 0.39
POLB P06746 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CSNK1D P48730 1/20 0.36
CSNK1E P49674 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HSP90AA1 P07900 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GPR35 Q9HC97 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205786 1.00 ALDH1A1 (0.50) ALDH1A1GSK3BGAATDP1PTGS1
SCHEMBL4482406 0.89 ALDH1A1 (0.42) ALDH1A1GSK3BGAATDP1PTGS1
SCHEMBL4482399 0.89 ALDH1A1 (0.42) ALDH1A1GSK3BGAATDP1PTGS1
SCHEMBL4479726 0.86 ALDH1A1 (0.50) ALDH1A1GSK3BGAATDP1TRPV1
SCHEMBL4479731 0.86 ALDH1A1 (0.50) ALDH1A1GSK3BGAATDP1TRPV1
SCHEMBL4485374 0.84 POLB (0.52) ALDH1A1GSK3BGAATDP1PTGS1
SCHEMBL4467387 0.84 POLB (0.52) ALDH1A1GSK3BGAATDP1PTGS1
SCHEMBL4469574 0.81 PTGS2 (0.51) ALDH1A1GSK3BTDP1PTGS1PTGS2
SCHEMBL4469564 0.81 PTGS2 (0.51) ALDH1A1GSK3BTDP1PTGS1PTGS2
SCHEMBL4464159 0.79 MAPT (0.45) ALDH1A1GSK3BGAATDP1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551842-A1 PYRADAZINE COMPOUNDS AS GSK-3 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-13 EP disclosed
WO-2004035588-A1 PYRADAZINE COMPOUNDS AS GSK-3 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-04-29 WO disclosed