SCHEMBL6205919

SCHEMBL6205919

Clc1cccc(Cl)c1COc1cnc(NCc2ccccc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 2/20 0.44
HPGD P15428 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPK1 P28482 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
GBA1 P04062 1/20 0.43
HDAC3 O15379 1/20 0.41
NCOR1 O75376 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
FABP1 P07148 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203080 0.80 KDM4E (0.41) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6238556 0.79 SMN1; SMN2 (0.44) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL6202806 0.76 PLK1 (0.40) MEN1KMT2ASMN1; SMN2POLBP2RX7
SCHEMBL6206177 0.71 SMN1; SMN2 (0.47) ALDH1A1KMT2APKMSMN1; SMN2KDM4E
SCHEMBL30723732 0.71 SMN1; SMN2 (0.47) ALDH1A1KMT2APKMSMN1; SMN2KDM4E
SCHEMBL6079114 0.70 SMN1; SMN2 (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL6078486 0.69 SMN1; SMN2 (0.41) HPGDKMT2AMAPK1CYP1A2CYP2C19
SCHEMBL6238555 0.69 SMN1; SMN2 (0.45) ALDH1A1KMT2APKMSMN1; SMN2KDM4E
SCHEMBL22191398 0.67 ALDH1A1 (0.57) ALDH1A1MEN1HPGDKMT2ACYP1A2
SCHEMBL6469221 0.67 MEN1 (0.57) ALDH1A1MEN1HPGDKMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545523-A1 3-&-grave;(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES ASP38 MAP KINASE INHIBITORS Astex Technology Limited (GB) 2005-06-29 EP disclosed
WO-2005002673-A1 RAF KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed
WO-2004004720-A1 3-`(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES AS P38 MAP KINASE INHIBITORS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO disclosed