SCHEMBL6206147

SCHEMBL6206147

Cc1nc2ncccc2cc1C(=O)N[C@H]1CC[C@H](C)CC1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
CNR2 P34972 18/20 0.56
CNR1 P21554 10/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206149 1.00 NPC1 (0.57) NPC1RAB9ACNR2CNR1
SCHEMBL6085332 0.78 CNR2 (0.58) NPC1RAB9ACNR2CNR1
SCHEMBL7736408 0.78 CNR2 (0.58) NPC1RAB9ACNR2CNR1
SCHEMBL6205946 0.76 RAB9A (0.51) NPC1RAB9ACNR2CNR1
SCHEMBL6205950 0.76 RAB9A (0.51) NPC1RAB9ACNR2CNR1
SCHEMBL12709415 0.75 P2RX7 (0.61) NPC1RAB9ACNR2CNR1
SCHEMBL7691769 0.75 EGLN1 (0.56) NPC1RAB9ACNR2CNR1
SCHEMBL125290 0.73 LMNA (0.51) NPC1RAB9A
SCHEMBL3458121 0.73 SMN1; SMN2 (0.53) NPC1RAB9A
SCHEMBL6085305 0.73 PLK1 (0.61) NPC1RAB9ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1595871-A2 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases NPS PHARMACEUTICALS, INC. (US) 2005-11-16 EP disclosed