SCHEMBL6206420

SCHEMBL6206420

COc1ncccc1-c1cocn1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.44
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
HRH4 Q9H3N8 1/20 0.40
CASP6 P55212 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ELANE P08246 1/20 0.39
CHRNA7 P36544 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
APLNR P35414 1/20 0.38
IMPDH2 P12268 3/20 0.38
KCNA3 P22001 1/20 0.38
DHODH Q02127 1/20 0.37
SCN9A Q15858 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
IMPDH1 P20839 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2122983 0.73 BTK (0.44) BTKNPC1RAB9AHRH4CA1
SCHEMBL16481976 0.71 BTK (0.42) BTKNPC1RAB9AHRH4CA1
SCHEMBL2121707 0.71 BTK (0.42) BTKNPC1RAB9AHRH4CA1
SCHEMBL27172748 0.71 IMPDH2 (0.39) NPC1RAB9AALOX5APFEN1IMPDH2
SCHEMBL26259970 0.70 SCN9A (0.47) NPC1CASP6IMPDH2SCN9AIMPDH1
SCHEMBL20801655 0.70 BTK (0.48) BTKNPC1RAB9AHRH4CA1
SCHEMBL12676837 0.70 BTK (0.48) BTKNPC1RAB9AHRH4CA1
SCHEMBL22939929 0.70 CCR1 (0.48) BTKNPC1RAB9AHRH4ELANE
SCHEMBL22940967 0.70 RAB9A (0.47) BTKNPC1RAB9AHRH4CASP6
SCHEMBL15344911 0.70 CCR1 (0.52) BTKNPC1RAB9AHRH4ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583749-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE Astellas Pharma Inc. (JP) 2005-10-12 EP disclosed
WO-2004065374-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE ASTELLAS PHARMA INC. (JP) 2004-08-05 WO disclosed