SCHEMBL6207384

SCHEMBL6207384

CC(=O)Nc1ccc2[nH]c(C(=O)N3CC(CCl)c4c3cc(N)c3ccccc43)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 2/20 0.44
ADH1A P07327 1/20 0.42
KIT P10721 1/20 0.42
FLT1 P17948 1/20 0.42
FLT4 P35916 1/20 0.42
KDR P35968 1/20 0.42
ABL2 P42684 1/20 0.42
MMP13 P45452 2/20 0.42
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
PYGL P06737 2/20 0.35
F11 P03951 2/20 0.34
MAOA P21397 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436370 0.92 MMP13 (0.46) HDAC2ADH1AKITFLT1FLT4
SCHEMBL6517367 0.92 ADH1A (0.52) HDAC2ADH1AKITFLT1FLT4
SCHEMBL6517373 0.92 ADH1A (0.52) HDAC2ADH1AKITFLT1FLT4
SCHEMBL10111775 0.88 MMP13 (0.42) HDAC2ADH1AKITFLT1FLT4
SCHEMBL469094 0.88 MMP13 (0.42) HDAC2ADH1AKITFLT1FLT4
SCHEMBL6204957 0.87 ADH1A (0.40) HDAC2ADH1AKITFLT1FLT4
SCHEMBL8107146 0.87 ADH1A (0.45) HDAC2ADH1AKITFLT1FLT4
SCHEMBL16151965 0.86 MMP13 (0.41) HDAC2ADH1AKITFLT1FLT4
SCHEMBL13498776 0.86 NPC1 (0.41) ADH1AKITFLT1FLT4KDR
SCHEMBL13800023 0.86 ADH1A (0.47) HDAC2ADH1AKITFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938474-B1 CYCLOPROPYLINDOLE COMPOUNDS AND THEIR USE AS PRODRUGS AUCKLAND UNISERVICES LTD (NZ) 2005-11-23 EP disclosed
US-6130237-A Condensed N-aclyindoles as antitumor agents CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-10-10 US disclosed