SCHEMBL6207417

SCHEMBL6207417

CCCCOC(=O)NC(CC(=O)O)c1nccs1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.55
PKM P14618 1/20 0.43
CTSA P10619 9/20 0.43
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 2/20 0.38
FAAH O00519 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201378 0.89 L3MBTL1 (0.54) L3MBTL1PKMCTSASMN1; SMN2NPC1
SCHEMBL2464521 0.77 L3MBTL1 (0.41) L3MBTL1SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL5086318 0.76 FAAH (0.45) L3MBTL1CTSASMN1; SMN2NPC1RAB9A
SCHEMBL3663114 0.76 L3MBTL1 (0.43) L3MBTL1SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL21552119 0.75 CTSA (0.45) CTSA
SCHEMBL21552487 0.75 CTSA (0.47) CTSA
SCHEMBL5504022 0.75 SMN1; SMN2 (0.42) L3MBTL1SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL14040614 0.75 SMN1; SMN2 (0.57) L3MBTL1SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL844472 0.75 SMN1; SMN2 (0.57) L3MBTL1SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL6207414 0.74 L3MBTL1 (0.55) L3MBTL1PKMSMN1; SMN2RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569954-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-09-07 EP disclosed
EP-1503997-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-02-09 EP disclosed
WO-2004052921-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-06-24 WO disclosed
WO-2003097617-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2003-11-27 WO disclosed