SCHEMBL5201378

SCHEMBL5201378

CCCCOC(=O)NC(CC(=O)OC)c1nccs1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.54
PKM P14618 1/20 0.43
RAB9A P51151 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 3/20 0.41
MAPK1 P28482 2/20 0.40
TSHR P16473 2/20 0.40
CYP3A4 P08684 1/20 0.39
FAAH O00519 1/20 0.37
CTSK P43235 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CTSA P10619 1/20 0.36
CASP1 P29466 1/20 0.36
HPGD P15428 1/20 0.36
PTPRB P23467 1/20 0.36
AGTR2 P50052 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207417 0.89 L3MBTL1 (0.55) L3MBTL1PKMRAB9ASMN1; SMN2NPC1
SCHEMBL4385673 0.74 SMN1; SMN2 (0.51) L3MBTL1RAB9ASMN1; SMN2NPC1MAPK1
SCHEMBL1721285 0.73 FAAH (0.47) L3MBTL1RAB9ASMN1; SMN2NPC1MAPK1
SCHEMBL5201374 0.73 L3MBTL1 (0.55) L3MBTL1PKMRAB9ASMN1; SMN2MAPK1
SCHEMBL4096169 0.72 POLB (0.51) L3MBTL1RAB9ASMN1; SMN2NPC1MAPK1
SCHEMBL3821977 0.71 MAPT (0.49) L3MBTL1PKMRAB9ASMN1; SMN2NPC1
SCHEMBL2345224 0.71 EPHX1 (0.42) L3MBTL1RAB9ASMN1; SMN2NPC1MAPK1
SCHEMBL11060290 0.71 EPHX1 (0.44) L3MBTL1RAB9ASMN1; SMN2NPC1MAPK1
SCHEMBL10809546 0.71 L3MBTL1 (1.00) L3MBTL1PKMRAB9ASMN1; SMN2NPC1
SCHEMBL6207414 0.71 L3MBTL1 (0.55) L3MBTL1PKMRAB9ASMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817275-A1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Schering Aktiengesellschaft (DE) 2007-08-15 EP disclosed
WO-2006060494-A1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2006-06-08 WO disclosed