SCHEMBL6207436

SCHEMBL6207436

COc1ccc(Nc2n[nH]c3cc(Cl)c(-c4ccccc4)cc23)cc1.Clc1cc2[nH]nc(Nc3ccccc3)c2cc1-c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.58
PRKAB2 O43741 5/20 0.56
PRKAG1 P54619 5/20 0.56
PRKAA2 P54646 5/20 0.56
PRKAA1 Q13131 5/20 0.56
PRKAG3 Q9UGI9 5/20 0.56
PRKAG2 Q9UGJ0 5/20 0.56
PRKAB1 Q9Y478 5/20 0.56
FADS1 O60427 1/20 0.55
CDK1 P06493 1/20 0.53
CDK2 P24941 1/20 0.53
PDGFRB P09619 2/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
CYP1A2 P05177 2/20 0.44
TRPA1 O75762 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPK10 P53779 1/20 0.43
MAPK14 Q16539 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4498877 0.99 PRKAB2 (0.57) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4503888 0.90 FADS1 (0.59) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4497901 0.89 GSK3B (0.70) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4495390 0.84 GSK3B (0.80) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4510158 0.84 GSK3B (0.60) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4498891 0.83 MAP2K4 (0.57) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4496233 0.81 PRKAB2 (0.65) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL27623023 0.81 MAPK8 (0.56) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4498900 0.81 TRPA1 (0.59) GSK3BPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4494950 0.80 TRPA1 (0.62) GSK3BFADS1CDK1CDK2ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537087-A1 NOVEL AMINOINDAZOLE DERIVATIVES AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Aventis Pharma S.A. (FR) 2005-06-08 EP disclosed
WO-2004022544-A1 NOVEL AMINOINDAZOLE DERIVATIVES AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AVENTIS PHARMA S.A. (FR) 2004-03-18 WO disclosed