SCHEMBL6207985

SCHEMBL6207985

COc1cc(-c2cc(COC(=O)C3CCNCC3)ccn2)cc(OC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 2/20 0.41
NEK2 P51955 4/20 0.41
TGFBR1 P36897 2/20 0.38
ACVR1 Q04771 2/20 0.38
ATM Q13315 2/20 0.38
FYN P06241 2/20 0.37
MAP3K11 Q16584 1/20 0.37
PLK1 P53350 1/20 0.37
NEK1 Q96PY6 1/20 0.37
ACVR1B P36896 1/20 0.37
KCNH2 Q12809 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FKBP1A P62942 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4122440 0.83 TGFBR1 (0.43) TGFBR1ACVR1FYNMAP3K11ACVR1B
SCHEMBL6168415 0.82 ALDH1A1 (0.55) ALDH1A1HPGDKCNH2SMN1; SMN2LMNA
SCHEMBL4122610 0.78 KDM4E (0.61) ALDH1A1KDM4EHPGDSMN1; SMN2KMT2A
SCHEMBL4127097 0.77 LMNA (0.40) ALDH1A1TGFBR1ACVR1MAP3K11ACVR1B
SCHEMBL4117314 0.76 KCNH2 (0.39) ALDH1A1TGFBR1ACVR1MAP3K11ACVR1B
SCHEMBL13813594 0.75 SLC6A2 (0.40) TGFBR1ACVR1FYNMAP3K11ACVR1B
SCHEMBL4108306 0.75 TGFBR1 (0.38) ALDH1A1KDM4ETGFBR1ACVR1MAP3K11
SCHEMBL4109512 0.75 SLC6A2 (0.41) ALDH1A1TGFBR1ACVR1MAP3K11ACVR1B
SCHEMBL4763695 0.73 CXCR4 (0.48) ALDH1A1KDM4ETGFBR1ACVR1ACVR1B
SCHEMBL6167568 0.73 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDKCNH2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494670-A1 MEDICINE FOR TREATING CANCER Kowa Co., Ltd. (JP) 2005-01-12 EP disclosed
WO-2003086397-A1 MEDICINE FOR TREATING CANCER KOWA CO., LTD. (JP) 2003-10-23 WO disclosed