SCHEMBL6208255

SCHEMBL6208255

NC(=O)N(c1ccccc1Br)c1ccc(CC(=O)O)cc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 4/20 0.41
AKR1B1 P15121 2/20 0.40
POLB P06746 2/20 0.39
LMNA P02545 2/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 2/20 0.39
ABCC4 O15439 1/20 0.39
PTGS1 P23219 1/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
RGS12 O14924 1/20 0.38
MAPT P10636 1/20 0.38
NFKB1 P19838 1/20 0.38
APEX1 P27695 1/20 0.38
THPO P40225 1/20 0.38
BLM P54132 1/20 0.38
GNAI1 P63096 1/20 0.38
PMP22 Q01453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6234919 0.86 GAA (0.48) NR3C1POLBLMNAGAATSHR
SCHEMBL6820924 0.84 AKR1B1 (0.41) NR3C1AKR1B1POLBLMNAGAA
SCHEMBL6825974 0.76 TRPA1 (0.39) MAPTALDH1A1
SCHEMBL6207117 0.74 CA2 (0.44) KDM4EHPGDHSD17B10RXRARXRB
SCHEMBL27516293 0.72 KDM4E (0.38) POLBLMNAGAATSHRKDM4E
SCHEMBL27499553 0.72 ACMSD (0.43) LMNAGAAHTTKDM4EHPGD
SCHEMBL5155305 0.72 GAA (0.49) LMNAGAATSHRPTGS1NFKB1
SCHEMBL6964628 0.72 GAA (0.46) POLBLMNAGAATSHRPTGS1
SCHEMBL27500465 0.71 HPGD (0.43) NR3C1LMNAHTTHPGDMAPT
SCHEMBL6962762 0.71 GAA (0.48) NR3C1LMNAGAATSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed