SCHEMBL6208323

SCHEMBL6208323

CN(C)CCOC(=O)N[CH]c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.49
BCHE P06276 4/20 0.48
ACHE P22303 2/20 0.45
ALDH1A1 P00352 3/20 0.44
CHRM2 P08172 2/20 0.43
CHRM3 P20309 2/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
POLB P06746 1/20 0.42
HRH1 P35367 1/20 0.42
LMNA P02545 1/20 0.42
CYP2D6 P10635 1/20 0.42
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4922122 0.83 LMNA (0.50) ALDH1A1POLBLMNAMEN1GAA
SCHEMBL3930322 0.80 TDP1 (0.58) ALDH1A1LMNAGAA
SCHEMBL4912299 0.79 MEN1 (0.54) ALDH1A1POLBLMNAMEN1GAA
SCHEMBL3934013 0.79 NPC1 (0.53) ALDH1A1LMNA
SCHEMBL14064867 0.77 CHRM1 (0.54) CHRM1BCHEALDH1A1CHRNB2CHRNA4
SCHEMBL9325467 0.76 BCHE (0.72) CHRM1BCHEALDH1A1LMNAMEN1
SCHEMBL3928127 0.76 LMNA (0.56) ALDH1A1POLBLMNAMEN1MAPT
SCHEMBL94681 0.75 ALDH1A1 (0.51) ALDH1A1LMNAGAAMAPT
SCHEMBL4023891 0.74 ALDH1A1 (0.72) BCHEACHEALDH1A1LMNAMEN1
SCHEMBL4023889 0.74 ALDH1A1 (0.72) BCHEACHEALDH1A1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383769-A4 6-SUBSTITUTED PYRAZOLO 3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2005-08-03 EP disclosed
EP-1383769-A2 6-SUBSTITUTED PYRAZOLO 3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS Bristol-Myers Squibb Pharma Company (US) 2004-01-28 EP disclosed
WO-2002067654-A3 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-10-31 WO disclosed
WO-2002067654-A2 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-09-06 WO disclosed