SCHEMBL6208564

SCHEMBL6208564

Cc1cc(COc2ccc(S(=O)(=O)CC(=O)C3CCNCC3)cc2)c2ccccc2n1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 19/20 0.65
MMP13 P45452 8/20 0.62
MMP2 P08253 2/20 0.56
MMP9 P14780 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3884532 0.89 ADAM17 (0.64) ADAM17MMP13MMP2MMP9
SCHEMBL6208690 0.88 ADAM17 (0.62) ADAM17MMP13MMP2
SCHEMBL6211162 0.84 MMP13 (0.64) ADAM17MMP13MMP2MMP9
SCHEMBL7107375 0.79 ADAM17 (1.00) ADAM17MMP13
SCHEMBL7106794 0.79 ADAM17 (1.00) ADAM17MMP13
SCHEMBL3860485 0.78 ADAM17 (0.75) ADAM17
SCHEMBL3860449 0.78 ADAM17 (0.75) ADAM17
SCHEMBL6208558 0.78 ADAM17 (0.59) ADAM17MMP13
SCHEMBL6100731 0.78 ADAM17 (0.67) ADAM17MMP13MMP2MMP9
SCHEMBL2681099 0.78 ADAM17 (0.67) ADAM17MMP13MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050256176-A1 Sulphonamide derivatives and their use as tace inhibitors ASTAZENECA AB (SE) 2005-11-17 US disclosed
EP-1539740-A1 SULPHONAMIDE DERIVATIVES AND THEIR USE AS TACE INHIBITORS AstraZeneca AB (SE) 2005-06-15 EP disclosed
WO-2004024715-A1 SULPHONAMIDE DERIVATIVES AND THEIR USE AS TACE INHIBITORS ASTRAZENECA AB (SE) 2004-03-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256176-A1 Sulphonamide derivatives and their use as tace inhibitors ADAM10, ADAM17, TNF ADAM17 2/4885MMP13 194/4885MMP2 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.