SCHEMBL6208619

SCHEMBL6208619

Nc1nc(NCCCc2c(-c3ccc(Cl)cc3Cl)c[nH]c2C(=O)OCc2ccccc2)ccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.46
GSK3A P49840 3/20 0.46
CDK1 P06493 2/20 0.46
CCNB2 O95067 1/20 0.46
CCNB1 P14635 1/20 0.46
CCNB3 Q8WWL7 1/20 0.46
SIRT5 Q9NXA8 3/20 0.38
PKM P14618 1/20 0.35
MAPT P10636 5/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR1 P21554 2/20 0.33
PLA2G1B P04054 1/20 0.32
ATG4B Q9Y4P1 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210081 0.88 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL13423054 0.81 GSK3B (0.46) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2903767 0.80 GSK3B (0.45) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL6429858 0.79 GSK3B (0.52) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL6213250 0.79 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL6408155 0.79 SIRT5 (0.41) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL6265338 0.77 GSK3B (0.48) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2912125 0.71 GSK3B (0.46) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2909753 0.71 HPGD (0.47) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2937412 0.71 GSK3B (0.46) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed