SCHEMBL6408155

SCHEMBL6408155

O=C(O)c1[nH]cc(-c2ccc(Cl)cc2Cl)c1CCCNc1ccc([N+](=O)[O-])c(Nc2ccccc2)n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 2/20 0.41
GSK3B P49841 6/20 0.39
GSK3A P49840 4/20 0.39
CDK1 P06493 2/20 0.39
CCNB2 O95067 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
STK17A Q9UEE5 1/20 0.36
PIN1 Q13526 1/20 0.36
FBP1 P09467 2/20 0.35
MAPT P10636 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
EIF4E P06730 1/20 0.34
FOLH1 Q04609 1/20 0.34
AURKA O14965 1/20 0.34
HSD11B1 P28845 1/20 0.33
KDM1A O60341 1/20 0.33
RCOR1 Q9UKL0 1/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210081 0.86 GSK3B (0.51) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL6208619 0.79 GSK3B (0.46) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL6408156 0.79 SIRT5 (0.39) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL6213250 0.75 GSK3B (0.51) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL6429858 0.74 GSK3B (0.52) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL6265338 0.68 GSK3B (0.48) SIRT5GSK3BGSK3ACDK1CCNB2
SCHEMBL29695661 0.66 GSK3B (0.61) GSK3BGSK3APIN1MAPTL3MBTL1
SCHEMBL7189543 0.65 GSK3B (0.56) SIRT5GSK3BGSK3APIN1MAPT
SCHEMBL7828769 0.65 SIRT5 (0.64) SIRT5STK17APIN1MAPTL3MBTL1
SCHEMBL6069007 0.65 GSK3B (0.53) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed