SCHEMBL6208735

SCHEMBL6208735

CSC(=O)c1ccc(C2CCCN2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.43
CHRNB2 P17787 2/20 0.41
CHRNA7 P36544 2/20 0.41
CHRNA4 P43681 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
PARP1 P09874 4/20 0.39
PARP2 Q9UGN5 2/20 0.39
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
MCHR1 Q99705 1/20 0.39
PARP3 Q9Y6F1 1/20 0.39
CHRM2 P08172 3/20 0.37
CHRM4 P08173 2/20 0.37
CHRM5 P08912 2/20 0.37
CHRM1 P11229 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21806659 0.82 MKNK1 (0.46) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL6208733 0.81 MKNK1 (0.40) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL28580499 0.80 PRKAB2 (0.48) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL3333833 0.79 PARP1 (0.50) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL13741356 0.78 ALDH1A1 (0.48) L3MBTL1SMN1; SMN2ALDH1A1MAPTPOLB
SCHEMBL4045684 0.78 MEN1 (0.45) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL38656217 0.76 PRKAB2 (0.51) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL38656590 0.76 PRKAB2 (0.51) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL38659922 0.76 PRKAB2 (0.51) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL16401323 0.76 KMT2A (0.46) MKNK1CHRNB2CHRNA7CHRNA4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed