SCHEMBL6208806

SCHEMBL6208806

COC(C(=O)O)=C(N)C(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
CES2 O00748 8/20 0.47
CES1 P23141 7/20 0.47
SRC P12931 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
MAPT P10636 3/20 0.43
POLB P06746 2/20 0.43
CYP3A4 P08684 1/20 0.43
PARP1 P09874 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 4/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.42
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208803 1.00 TSHR (0.48) TSHRCES2CES1SRCL3MBTL1
SCHEMBL6208814 0.87 TSHR (0.50) TSHRCES2CES1SRCL3MBTL1
SCHEMBL27923392 0.81 TSHR (0.52) TSHRCES2CES1SRCL3MBTL1
SCHEMBL6206511 0.81 ALDH1A1 (0.53) TSHRCES2CES1L3MBTL1MAPT
SCHEMBL27589200 0.78 TSHR (0.48) TSHRCES2CES1SRCL3MBTL1
SCHEMBL6576791 0.76 TSHR (0.56) TSHRCES2CES1SRCL3MBTL1
SCHEMBL6205114 0.75 CES2 (0.56) TSHRCES2CES1L3MBTL1MAPT
SCHEMBL8844091 0.75 CES2 (0.56) TSHRCES2CES1SRCL3MBTL1
SCHEMBL6205110 0.75 CES2 (0.56) TSHRCES2CES1L3MBTL1MAPT
SCHEMBL457034 0.75 TSHR (0.54) TSHRCES2CES1SRCL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532128-A1 INHIBITORS OF HCV NS5B POLYMERASE Pharmacia & Upjohn Company LLC (US) 2005-05-25 EP disclosed
WO-2004002977-A1 INHIBITORS OF HCV NS5B POLYMERASE PHARMACIA & UPJOHN COMPANY LLC (US) 2004-01-08 WO disclosed