SCHEMBL6208831

SCHEMBL6208831

CCOC(=O)CN1CCN(CCBr)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
TRPA1 O75762 1/20 0.45
GSK3B P49841 3/20 0.40
GSK3A P49840 2/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
ELANE P08246 1/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.37
MAPK1 P28482 1/20 0.37
HTR1A P08908 1/20 0.36
HTR2C P28335 1/20 0.36
PKM P14618 1/20 0.36
PIN1 Q13526 1/20 0.36
PIN4 Q9Y237 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912811 0.87 MGAM (0.50) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL11852921 0.87
SCHEMBL2373233 0.87 MGAM (0.50) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL3966571 0.87 MGAM (0.50) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL13296281 0.85 GSK3A (0.42) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL5153472 0.84 GSK3A (0.41) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL1127888 0.83 ALDH1A1 (0.45) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL21383465 0.83 HRH2 (0.41) ALDH1A1GSK3BGSK3APOLB
SCHEMBL4469979 0.82 ALOX15 (0.46) ALDH1A1TRPA1GSK3BGSK3AMGAM
SCHEMBL13612616 0.82 HRH2 (0.40) GSK3BGSK3AMGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed