SCHEMBL6208835

SCHEMBL6208835

N=C(N)c1cccc(C(F)(F)F)c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
KLK1 P06870 2/20 0.37
KLK5 Q9Y337 2/20 0.37
PTGS1 P23219 1/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
F10 P00742 1/20 0.35
PARP1 P09874 2/20 0.35
CA2 P00918 1/20 0.34
GRIN2D O15399 2/20 0.34
GRIN3B O60391 2/20 0.34
GRIN1 Q05586 2/20 0.34
GRIN2A Q12879 2/20 0.34
GRIN2B Q13224 2/20 0.34
GRIN2C Q14957 2/20 0.34
GRIN3A Q8TCU5 2/20 0.34
TAS2R14 Q9NYV8 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26135741 0.82 LMNA (0.39) LMNAGAAPTGS1KCNK3KCNK9
SCHEMBL29712527 0.82 LMNA (0.50) LMNAGAAPTGS1KCNK3KCNK9
SCHEMBL958496 0.82 LMNA (0.50) LMNAGAAPTGS1KCNK3KCNK9
SCHEMBL8513460 0.81 PARP1 (0.47) LMNAGAAPTGS1KCNK3KCNK9
Hydrochloric Acid SCHEMBL3065338 0.80 LMNA (0.48) LMNAGAAPTGS1F10GRIN2D
Hydrochloric Acid SCHEMBL31138645 0.80 LMNA (0.48) LMNAGAAPTGS1F10GRIN2D
Hydrochloric Acid SCHEMBL27788451 0.79 LMNA (0.37) LMNAGAAPTGS1CTSSCTSK
Hydrochloric Acid SCHEMBL1259553 0.78 LMNA (0.47) LMNAGAAPTGS1GRIN2DGRIN3B
SCHEMBL396017 0.76 CA2 (0.55) LMNAGAACA2ALDH1A1POLB
SCHEMBL28052029 0.76 LMNA (0.48) LMNAGAAPTGS1KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014062938-A1 RORY MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2014-04-24 WO disclosed
CN-101115482-A Heterocyclic aspartyl protease inhibitors SCHERING CORP (US) 2008-01-30 CN disclosed
EP-1458392-A4 ACRIDONE INHIBITORS OF IMPDH ENZYME BRISTOL MYERS SQUIBB CO (US) 2005-06-08 EP disclosed
EP-1458392-A2 ACRIDONE INHIBITORS OF IMPDH ENZYME Bristol-Myers Squibb Company (US) 2004-09-22 EP disclosed
WO-2003059269-A2 ACRIDONE INHIBITORS OF IMPDH ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-24 WO disclosed