SCHEMBL6208886

SCHEMBL6208886

Cc1cccc(N(Br)C(=O)NOC(=O)Cc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.47
RAB9A P51151 5/20 0.43
NPC1 O15118 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HTT P42858 2/20 0.43
JAK2 O60674 1/20 0.43
PAX8 Q06710 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 1/20 0.38
POLB P06746 1/20 0.37
RECQL P46063 1/20 0.37
LMNA P02545 1/20 0.37
HSP90AA1 P07900 1/20 0.37
PTGIR P43119 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6209618 0.85 L3MBTL1 (0.47) L3MBTL1RAB9ANPC1ALDH1A1HTT
SCHEMBL6208199 0.77 PTGS1 (0.40) RAB9ANPC1ALDH1A1HTTJAK2
SCHEMBL5156830 0.75 TSHR (0.47) L3MBTL1RAB9AALDH1A1SMN1; SMN2TDP1
SCHEMBL6208226 0.74 KMT2A (0.56) L3MBTL1RAB9ANPC1ALDH1A1KMT2A
SCHEMBL5152783 0.73 L3MBTL1 (0.44) L3MBTL1ALDH1A1HTTKMT2AMEN1
SCHEMBL6208938 0.72 CNR2 (0.41) RAB9AKMT2AMEN1SMN1; SMN2TSHR
SCHEMBL1704086 0.70 RAB9A (0.49) RAB9ANPC1ALDH1A1HTTJAK2
SCHEMBL27516923 0.69 TSHR (0.53) L3MBTL1ALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL29393816 0.68 SMN1; SMN2 (0.61) L3MBTL1ALDH1A1HTTKMT2AMEN1
SCHEMBL1640435 0.68 SMN1; SMN2 (0.61) L3MBTL1ALDH1A1HTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed