Carbromal

Carbromal

SCHEMBL620919

CCC(Br)(CC)C(=O)NC(N)=O.O=P(O)(O)O

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Carbromal. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.33
NR3C1 P04150 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbromal SCHEMBL1537493 0.98 CRBN (0.32) CRBN
Carbromal SCHEMBL4183308 0.94 CRBN (0.32) CRBN
Carbromal SCHEMBL11114786 0.93
Carbromal SCHEMBL1499641 0.93 SLC34A1 (0.32) CRBN
Carbromal SCHEMBL15057476 0.92 CRBN (0.39) CRBNNR3C1
Carbromal SCHEMBL261 0.92 CRBN (0.39) CRBNNR3C1
Carbromal SCHEMBL4351621 0.92 CRBN (0.39) CRBNNR3C1
Carbromal SCHEMBL11332793 0.91 CRBN (0.30) CRBN
Carbromal SCHEMBL8594411 0.91 MMP1 (0.32) CRBN
Carbromal SCHEMBL10866938 0.91 SLC34A1 (0.31) CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230072480-A1 COVALENT FUNCTIONALIZATION OF GRAPHENE UNIVERSIDAD REY JUAN CARLOS (ES) 2023-03-09 US claimed
EP-4105176-A1 COVALENT FUNCTIONALISATION OF GRAPHENE Universidad Rey Juan Carlos (ES) 2022-12-21 EP claimed
WO-2021160911-A1 COVALENT FUNCTIONALISATION OF GRAPHENE UNIVERSIDAD REY JUAN CARLOS (ES) 2021-08-19 WO claimed
US-20110070347-A1 COMPOSITION FOR BLOCKING INTERFIBRILLAR SPACES IN MEAT AND MEAT TREATMENT METHODS USING SAID COMPOSITION TECNOALIMENTICA LTDA 2011-03-24 US claimed
WO-2002085136-A2 MIXTURE FOR IMPROVING THE COOKING MEAT PRODUCTS AND PROCESS FOR ITS USE TECNOALIMENTICA LTDA (CO) 2002-10-31 WO claimed
EP-0780463-B1 High load-carrying lubricating oils containing amine phosphate and thiophene carboxylic acid derivatives BP PRODUCTS NORTH AMERICA INC (US) 2002-08-07 EP claimed
EP-0780462-B1 High load-carrying turbo oils containing amine phosphate and a sulfur containing carboxylic acid BP EXPLORATION AND OIL INC (US) 2001-07-25 EP claimed
US-5750478-A High load-carrying turbo oils containing amine phosphate and sulfurized fatty acid EXXON RESEARCH AND ENGINEERING COMPANY (US) 1998-05-12 US claimed
US-5679627-A ADIITIVE MIXTURE OF SULFUR CONTAINING CARBOXYLIC ACIDS AND ONE OR MORE AMINE PHOSPHATES EXXON RESEARCH & ENGINEERING COMPANY (US) 1997-10-21 US claimed
US-5587355-A SYNERGISTIC MIXTURE IMPROVES WEAR RESISTANCE EXXON RESEARCH AND ENGINEERING COMPANY (US) 1996-12-24 US claimed
US-5585029-A STABILIZERS; SYNERGISTIC, WEAR RESISTANCE EXXON RESEARCH AND ENGINEERING COMPANY (US) 1996-12-17 US claimed
US-5582760-A POLYOL ESTER BASED TURBINE OIL; OXIDATION AND CORROSION RESISTANCE, SILICON SEAL COMPATIBILITY EXXON RESEARCH AND ENGINEERING COMPANY (US) 1996-12-10 US claimed
US-4716034-A POLYETHYLENE OXIDE STABILIZER AGAINST SYNERESIS COLGATE-PALMOLIVE COMPANY (US) 1987-12-29 US claimed
US-4716036-A PREVENTION OF SYNERESIS FROM CONTACT WITH POLYOLEFIN COLGATE-PALMOLIVE COMPANY (US) 1987-12-29 US claimed
US-4021230-A AMMONIUM IMINES AMCHEM PRODUCTS, INC. (US) 1977-05-03 US claimed
US-4007128-A GELLED HYDROCARBON BORG-WARNER CORPORATION (US) 1977-02-08 US claimed
JP-5125049-A None JP disclosed
CN-111662330-B Substituted 4-phenylpyridines for the treatment of NK-1 receptor related diseases 赫尔森保健股份公司 2023-05-12 CN disclosed
US-4021230-A AMMONIUM IMINES AMCHEM PRODUCTS, INC. (US) 1977-05-03 US disclosed
US-3970238-A FLUX OF PHOSPHOROUS OR PHOSPHORIC ACID AND PHOSPHATE SALTS LAKE CHEMICAL COMPANY (US) 1976-07-20 US disclosed