SCHEMBL6209230

SCHEMBL6209230

CCCC(NC(=O)c1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.45
HTRA1 Q92743 1/20 0.43
DRD4 P21917 1/20 0.43
MC4R P32245 2/20 0.41
MC3R P41968 2/20 0.41
MC1R Q01726 2/20 0.41
GPR132 Q9UNW8 3/20 0.40
CTSK P43235 3/20 0.40
SMYD3 Q9H7B4 2/20 0.38
ACE P12821 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
AKT1 P31749 1/20 0.36
PTAFR P25105 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041827 0.90 CTSK (0.43) CCR1HTRA1GPR132CTSKSMYD3
SCHEMBL4040649 0.90 CTSK (0.42) CCR1GPR132CTSKSMYD3ACE
SCHEMBL4039411 0.90 CTSK (0.43) CCR1GPR132CTSKACE
SCHEMBL4042695 0.90 CHRNB2 (0.41) GPR132CTSKPTAFR
SCHEMBL4047844 0.89 SMYD3 (0.35) HTRA1DRD4MC4RMC3RMC1R
SCHEMBL6211183 0.89 CTSK (0.42) HTRA1MC4RMC3RMC1RCTSK
SCHEMBL4045831 0.89 CTSK (0.51) GPR132CTSKSMYD3ACE
SCHEMBL4042752 0.88 CTSK (0.52) GPR132CTSKSMYD3ACE
SCHEMBL4038224 0.88 CTSK (0.44) GPR132CTSKSMYD3ACETAAR1
SCHEMBL6210263 0.88 CTSK (0.44) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed