SCHEMBL6209260

SCHEMBL6209260

Nc1cc(F)c(N2CC3OC3C2)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.34
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
GFER P55789 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18396703 0.81 MTOR (0.36) MAOA
SCHEMBL240100 0.81 KDM4E (0.46) MAOAALDH1A1LMNAMAPTTDP1
SCHEMBL29209046 0.81 KDM4E (0.46) MAOAALDH1A1LMNAMAPTTDP1
SCHEMBL4706606 0.80 MAOA (0.33) MAOAALDH1A1LMNAMAPTMAPK1
SCHEMBL239087 0.78 MAOA (0.32) MAOAALDH1A1LMNAMAPTMAPK1
SCHEMBL238837 0.78 MAOA (0.32) MAOAALDH1A1LMNAMAPTMAPK1
SCHEMBL241355 0.76 ALDH1A1 (0.32) MAOAALDH1A1
SCHEMBL236762 0.76 KDM4E (0.35) MAOAALDH1A1MAPT
SCHEMBL241891 0.76 ALDH1A1 (0.32) MAOAALDH1A1
SCHEMBL22698326 0.75 MAOA (0.35) MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1549641-A1 ANTIMICROBIAL 3.1.0 BICYCLIC OXAZOLIDINONE DERIVATIVES Pharmacia & Upjohn Company LLC (US) 2005-07-06 EP disclosed
US-6875784-B2 Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives PHARMACIA & UPJOHN COMPANY (US) 2005-04-05 US disclosed
US-20040127530-A1 Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives PHARMACIA & UPJOHN COMPANY 2004-07-01 US disclosed
WO-2004033451-A1 ANTIMICROBIAL [3.1.0] BICYCLIC OXAZOLIDINONE DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127530-A1 Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives OXA1L, CYP1B1, MT-CO1 MAOA 743/4885ALDH1A1 345/4885LMNA 2200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.