SCHEMBL6209566

SCHEMBL6209566

C=CC(c1ccccc1)C1C(=O)OC(C)(c2ccccc2)C(=O)C1=O

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CYP1A2 P05177 1/20 0.33
EGFR P00533 1/20 0.31
ALDH1A1 P00352 1/20 0.31
DHODH Q02127 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6175595 0.76 EGFR (0.35) EGFRALDH1A1
SCHEMBL28548234 0.61 HCAR2 (0.53) HCAR3HCAR2CYP1A2ALDH1A1DHODH
SCHEMBL17070911 0.60 ALDH1A1 (0.40) CYP1A2ALDH1A1
SCHEMBL6843663 0.60 MEN1 (0.41) CYP1A2ALDH1A1
SCHEMBL13716378 0.59 CYP1A2 (0.45) HCAR3HCAR2CYP1A2ALDH1A1DHODH
SCHEMBL4352151 0.58 CA2 (0.42) HCAR3HCAR2CYP1A2ALDH1A1DHODH
SCHEMBL1690392 0.58 CHRM2 (0.37)
SCHEMBL5679073 0.57 MAPT (0.33) ALDH1A1
SCHEMBL2804521 0.57 ALDH1A1 (0.37) CYP1A2ALDH1A1
SCHEMBL23214499 0.56 HCAR2 (0.45) HCAR3HCAR2CYP1A2EGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP claimed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed