SCHEMBL6209893

SCHEMBL6209893

CCc1ccc(-c2c[nH]c(CCCNc3ccc([N+](=O)[O-])c(N)n3)c2NC(=O)CNCCCOC)cc1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC1 Q13547 1/20 0.31
GSK3A P49840 2/20 0.30
GSK3B P49841 2/20 0.30
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211337 0.85 GSK3A (0.33) MAPK1GSK3AGSK3BCCNB2CDK1
SCHEMBL2911941 0.82 HDAC1 (0.34) ALDH1A1MAPK1KMT2AHDAC1GSK3A
SCHEMBL2909547 0.80 GSK3B (0.37) GSK3AGSK3BCCNB2CDK1CCNB1
Hydrochloric Acid SCHEMBL2911853 0.80 KAT2B (0.37) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL6270770 0.78 BCL2 (0.34)
SCHEMBL2912926 0.72 BDKRB1 (0.34) KMT2AGSK3AGSK3B
SCHEMBL2905411 0.69 GSK3B (0.35) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL2907410 0.69 GSK3B (0.34) ALDH1A1MAPK1KMT2AGSK3AGSK3B
SCHEMBL2912527 0.69 GSK3B (0.36) KMT2AGSK3AGSK3BCDK1
SCHEMBL2908407 0.68 GSK3B (0.34) GSK3AGSK3BCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed