SCHEMBL6270770

SCHEMBL6270770

CCc1ccc(-c2c[nH]c(CCCNc3ccc([N+](=O)[O-])c(N)n3)c2NC(=O)C(COC(C)(C)C)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 6/20 0.34
GSTP1 P09211 1/20 0.32
GSTM2 P28161 1/20 0.32
MCL1 Q07820 1/20 0.32
SCN9A Q15858 2/20 0.31
ACHE P22303 1/20 0.31
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211337 0.90 GSK3A (0.33) BCL2
SCHEMBL2909660 0.84 BCL2 (0.33) BCL2GSTP1GSTM2MCL1SCN9A
SCHEMBL6209893 0.78 ALDH1A1 (0.32)
SCHEMBL2909547 0.78 GSK3B (0.37)
Hydrochloric Acid SCHEMBL2911853 0.77 KAT2B (0.37)
SCHEMBL2907603 0.75 CA2 (0.35) BCL2
SCHEMBL2912738 0.74 BCL2 (0.32) BCL2GSTP1GSTM2MCL1SCN9A
SCHEMBL2907410 0.73 GSK3B (0.34)
SCHEMBL2907714 0.71 GSK3B (0.42) BCL2GSTP1GSTM2MCL1
SCHEMBL2905411 0.70 GSK3B (0.35) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed