SCHEMBL6211337

SCHEMBL6211337

CCc1ccc(-c2c[nH]c(CCCNc3ccc([N+](=O)[O-])c(N)n3)c2NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
SIRT5 Q9NXA8 1/20 0.31
KAT2B Q92831 1/20 0.31
CYP17A1 P05093 1/20 0.31
BCL2 P10415 1/20 0.30
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
ABCB11 O95342 1/20 0.30
ESR1 P03372 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6270770 0.90 BCL2 (0.34) BCL2
SCHEMBL6209893 0.85 ALDH1A1 (0.32) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL2909547 0.84 GSK3B (0.37) GSK3AGSK3BCCNB2CDK1CCNB1
Hydrochloric Acid SCHEMBL2911853 0.84 KAT2B (0.37) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL2907410 0.80 GSK3B (0.34) GSK3AGSK3BCDK1KAT2BCYP17A1
SCHEMBL6209689 0.78 CYP17A1 (0.38) CYP17A1
SCHEMBL2905411 0.76 GSK3B (0.35) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL8041119 0.74 STK17B (0.46) SIRT5
SCHEMBL6265338 0.74 GSK3B (0.48) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL2909660 0.72 BCL2 (0.33) BCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed