SCHEMBL6209898

SCHEMBL6209898

CCN(CC)c1ccc(C(=O)NCCC(C)CC(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2ccccn2)cc1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.38
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 1/20 0.36
CTSL P07711 13/20 0.36
CTSS P25774 12/20 0.36
ELOVL6 Q9H5J4 1/20 0.35
CTSV O60911 1/20 0.34
CTSB P07858 1/20 0.34
SMYD3 Q9H7B4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210934 0.94 CTSK (0.44) CTSKGAACTSLCTSSCTSV
SCHEMBL6210259 0.91 MEN1 (0.38) CTSKCTSLCTSSCTSVCTSB
SCHEMBL6211016 0.91 CTSK (0.37) CTSKCTSLCTSSCTSVCTSB
SCHEMBL6213254 0.90 CTSK (0.44) CTSKALDH1A1CTSLCTSSCTSV
SCHEMBL6211626 0.89 CCR5 (0.38) CTSKCTSLCTSS
SCHEMBL6211360 0.89 CHRM4 (0.40) CTSKALDH1A1GAACTSLCTSS
SCHEMBL6213978 0.89 CASR (0.38) CTSKCTSLCTSSCTSVCTSB
SCHEMBL6210002 0.89 CTSK (0.36) CTSKCTSLCTSSCTSVCTSB
SCHEMBL6211873 0.88 CTSK (0.39) CTSKCTSLCTSS
SCHEMBL6209035 0.88 CTSK (0.36) CTSKALDH1A1SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed