SCHEMBL6213751

SCHEMBL6213751

c1cnc(Oc2cccc3ccccc23)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
HPGD P15428 3/20 0.50
MAPT P10636 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50
HTR1B P28222 5/20 0.47
KDM4E B2RXH2 4/20 0.44
KCNA3 P22001 1/20 0.44
NISCH Q9Y2I1 1/20 0.44
GAA P10253 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HTR1D P28221 1/20 0.43
CYP3A4 P08684 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9858926 0.85 SIRT2 (0.47) ALDH1A1HPGDMAPTTDP1MEN1
SCHEMBL5733557 0.81 KDM4E (0.67) ALDH1A1HPGDMAPTTDP1MEN1
SCHEMBL11133778 0.80 MEN1 (0.48) ALDH1A1MAPTMEN1NPC1POLB
SCHEMBL442767 0.80 HTR1B (0.54) ALDH1A1HPGDMAPTTDP1MEN1
SCHEMBL29577853 0.80 HTR1B (0.54) ALDH1A1HPGDMAPTTDP1MEN1
SCHEMBL1884690 0.79 TRPA1 (0.48) ALDH1A1HPGDMAPTTDP1MEN1
Methane SCHEMBL10959030 0.78 HTR1B (0.52) ALDH1A1HPGDMAPTTDP1MEN1
Lithium SCHEMBL6571336 0.78 HTR1B (0.52) ALDH1A1HPGDMAPTTDP1MEN1
SCHEMBL7457103 0.78 HTR1B (0.52) ALDH1A1HPGDMAPTTDP1MEN1
Phosphine SCHEMBL28264511 0.78 HTR1B (0.52) ALDH1A1HPGDMAPTTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224183-B1 HETEROCYCLIC SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL MYERS SQUIBB CO (US) 2005-12-28 EP claimed