SCHEMBL6217477

SCHEMBL6217477

Nc1nc(-c2c[c]ccc2)cs1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.62
CYP3A4 P08684 2/20 0.62
RAB9A P51151 8/20 0.58
MAPT P10636 7/20 0.58
NPC1 O15118 7/20 0.58
KDM4E B2RXH2 4/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
NFKB1 P19838 2/20 0.58
NFKB2 Q00653 2/20 0.58
RELA Q04206 2/20 0.58
LMNA P02545 1/20 0.58
HPGD P15428 1/20 0.51
HK1 P19367 1/20 0.51
HKDC1 Q2TB90 1/20 0.51
LTA4H P09960 4/20 0.49
AR P10275 1/20 0.49
GFER P55789 1/20 0.49
MKNK1 Q9BUB5 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3801938 0.84 KDM4E (0.51) ALDH1A1RAB9AMAPTNPC1KDM4E
SCHEMBL9957782 0.81 KDM4E (0.62) ALDH1A1CYP3A4RAB9AMAPTNPC1
SCHEMBL61174 0.81 RECQL (0.53) ALDH1A1RAB9AMAPTNPC1KDM4E
Hydrochloric Acid SCHEMBL5450269 0.77 ALDH1A1 (0.92) ALDH1A1CYP3A4RAB9AMAPTNPC1
Bromide SCHEMBL5325472 0.77 ALDH1A1 (1.00) ALDH1A1CYP3A4RAB9AMAPTNPC1
SCHEMBL1029102 0.77 ALDH1A1 (0.66) ALDH1A1CYP3A4RAB9AMAPTNPC1
SCHEMBL44869 0.77 ALDH1A1 (1.00) ALDH1A1CYP3A4RAB9AMAPTNPC1
Bromide SCHEMBL7128948 0.75 ALDH1A1 (0.96) ALDH1A1CYP3A4RAB9AMAPTNPC1
SCHEMBL1771825 0.74 ALDH1A1 (0.79) ALDH1A1CYP3A4RAB9AMAPTNPC1
SCHEMBL2907964 0.73 ALDH1A1 (1.00) ALDH1A1CYP3A4RAB9AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1587800-A1 THIAZOLE DERIVATIVES AND THEIR USE AS VAP-1 INHIBITORS Astellas Pharma Inc. (JP) 2005-10-26 EP disclosed
WO-2004067521-A1 THIAZOLE DERIVATIVES AND THEIR USE AS VAP-1 INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-08-12 WO disclosed