SCHEMBL6220199

SCHEMBL6220199

O=C(O)c1ccc(-c2ccc(NCc3ccc4c(c3)OCCO4)cn2)s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.64
POLB P06746 1/20 0.43
BRAF P15056 1/20 0.43
GAA P10253 4/20 0.43
ALDH1A1 P00352 3/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 1/20 0.43
MAPT P10636 4/20 0.42
MEN1 O00255 2/20 0.42
ALOX15 P16050 2/20 0.42
KMT2A Q03164 2/20 0.42
VNN1 O95497 1/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
P4HTM Q9NXG6 1/20 0.41
CYP3A4 P08684 2/20 0.41
HDAC3 O15379 2/20 0.41
HDAC2 Q92769 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5904070 0.91 HDAC1 (0.61) HDAC1POLBBRAFGAAALDH1A1
SCHEMBL5903893 0.91 HDAC1 (0.78) HDAC1MEN1KMT2ACYP3A4HDAC3
SCHEMBL6197819 0.72 HDAC1 (0.60) HDAC1CYP3A4HDAC3HDAC2HDAC6
SCHEMBL6529911 0.71 HDAC1 (0.64) HDAC1CYP3A4HDAC3HDAC2HDAC6
SCHEMBL6246675 0.70 HDAC6 (0.72) HDAC1POLBGAAALDH1A1HSD17B10
SCHEMBL11230733 0.69 ALDH1A1 (0.70) HDAC1GAAALDH1A1HSD17B10KDM4E
SCHEMBL5903852 0.69 HDAC1 (0.58) HDAC1ALDH1A1KDM4EL3MBTL1MEN1
SCHEMBL11426003 0.68 ALDH1A1 (0.68) HDAC1GAAALDH1A1HSD17B10KDM4E
SCHEMBL9335999 0.68 MAPT (0.50) POLBALDH1A1HSD17B10KDM4EL3MBTL1
SCHEMBL5903880 0.67 HDAC1 (0.84) HDAC1KDM4EMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1525199-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS AS HISTONE DEACETYLASE INHIBITORS Argenta Discovery Limited (GB) 2005-04-27 EP claimed
WO-2004013130-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS AS HISTONE DEACETYLASE INHIBITORS ARGENTA DISCOVERY LIMITED (GB) 2004-02-12 WO claimed