SCHEMBL6220929

SCHEMBL6220929

NC(=O)[C@@H]1CCN(Cc2cc3c(N)ncnc3s2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.35
LIMK1 P53667 1/20 0.35
ADORA2A P29274 9/20 0.35
ADORA1 P30542 7/20 0.34
DGAT1 O75907 1/20 0.34
P2RY12 Q9H244 3/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7213496 0.93 P2RY12 (0.35) MEN1ADORA2AADORA1DGAT1P2RY12
SCHEMBL7213537 0.88 SELE (0.44) MEN1P2RY12KMT2A
SCHEMBL6220931 0.84 ADORA2A (0.36) MEN1ADORA2AADORA1KMT2A
SCHEMBL6221794 0.83 SIRT2 (0.38) DGAT1
Hydrochloric Acid SCHEMBL6435657 0.81 F10 (0.38) ADORA2AADORA1
Trifluoroacetic Acid SCHEMBL7213497 0.81 P2RY12 (0.36) MEN1ADORA2AADORA1DGAT1P2RY12
Trifluoroacetic Acid SCHEMBL6221816 0.78 SIRT2 (0.35) MEN1DGAT1
SCHEMBL6221508 0.76 F10 (0.49) DGAT1
SCHEMBL7213538 0.72 SELE (0.48) MEN1ADORA2AADORA1KMT2A
SCHEMBL1652680 0.72 F10 (0.34) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086099-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2005-09-28 EP claimed
EP-1086099-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2005-09-28 EP disclosed