SCHEMBL7213538

SCHEMBL7213538

N[C@H]1CCN(Cc2cc3c(Cl)ncnc3s2)C1=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SELE P16581 1/20 0.48
VCAM1 P19320 1/20 0.48
MEN1 O00255 12/20 0.35
KMT2A Q03164 9/20 0.35
KDM4E B2RXH2 2/20 0.34
HRH4 Q9H3N8 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HTT P42858 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
F10 P00742 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6220931 0.87 ADORA2A (0.36) MEN1KMT2AKDM4EHRH4ALDH1A1
SCHEMBL7213537 0.84 SELE (0.44) SELEVCAM1MEN1KMT2AKDM4E
SCHEMBL27502979 0.81 SELE (0.46) SELEVCAM1MEN1KMT2AKDM4E
SCHEMBL7215808 0.81 F10 (0.47) ADORA2AADORA1F10
Hydrochloric Acid SCHEMBL7219453 0.80 F10 (0.47) ADORA2AADORA1F10
Hydrochloric Acid SCHEMBL7219449 0.80 F10 (0.47) ADORA2AADORA1F10
Trifluoroacetic Acid SCHEMBL7213497 0.79 P2RY12 (0.36) MEN1KMT2AADORA2AADORA1
SCHEMBL27504720 0.77 SELE (0.39) SELEVCAM1MEN1KMT2AHDAC3
SCHEMBL7213522 0.75 SELE (0.40) SELEVCAM1MEN1KMT2AHDAC3
SCHEMBL7448973 0.75 SELE (0.40) SELEVCAM1MEN1KMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602864-B1 Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-08-05 US disclosed
EP-0944386-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6281227-B1 INHIBITORS OF THE ACTIVITY OF FACTOR XA. AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-08-28 US disclosed