SCHEMBL7213537

SCHEMBL7213537

NC(=O)[C@@H]1CCN(Cc2cc3c(Cl)ncnc3s2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SELE P16581 1/20 0.44
VCAM1 P19320 1/20 0.44
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
F10 P00742 2/20 0.35
MEN1 O00255 11/20 0.35
KMT2A Q03164 5/20 0.33
F2 P00734 1/20 0.33
PLG P00747 1/20 0.33
PLAT P00750 1/20 0.33
PROC P04070 1/20 0.33
P2RY12 Q9H244 3/20 0.33
JAK3 P52333 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6220929 0.88 MEN1 (0.35) MEN1KMT2AP2RY12
SCHEMBL7213538 0.84 SELE (0.48) SELEVCAM1HDAC3HDAC1HDAC6
Trifluoroacetic Acid SCHEMBL7213496 0.82 P2RY12 (0.35) MEN1KMT2AP2RY12
SCHEMBL27502979 0.80 SELE (0.46) SELEVCAM1HDAC3HDAC1HDAC6
SCHEMBL27504720 0.79 SELE (0.39) SELEVCAM1HDAC3HDAC1HDAC6
SCHEMBL7452311 0.77 CNR1 (0.38) F10JAK3ALDH1A1
SCHEMBL7219969 0.77 CNR1 (0.38) F10JAK3ALDH1A1
SCHEMBL6221794 0.76 SIRT2 (0.38)
SCHEMBL7213522 0.76 SELE (0.40) SELEVCAM1HDAC3HDAC1HDAC6
SCHEMBL7448973 0.76 SELE (0.40) SELEVCAM1HDAC3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602864-B1 Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-08-05 US disclosed
EP-0944386-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6281227-B1 INHIBITORS OF THE ACTIVITY OF FACTOR XA. AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-08-28 US disclosed
WO-2001039759-A2 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-06-07 WO disclosed