SCHEMBL622672

SCHEMBL622672

Oc1ccc2ccc(Cl)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
ESR2 Q92731 8/20 0.41
HSD17B10 Q99714 1/20 0.41
TTR P02766 2/20 0.41
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
ENPP2 Q13822 1/20 0.40
ESR1 P03372 7/20 0.40
CYP1A2 P05177 1/20 0.39
ESRRB O95718 1/20 0.38
ESRRA P11474 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL483970 0.84 ESR2 (0.55) ALDH1A1MEN1KMT2ACASP1CASP7
Hydrochloric Acid SCHEMBL7794275 0.83 ESR2 (0.53) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL20480300 0.82 MEN1 (0.37) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL20480301 0.82 MEN1 (0.37) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL25284715 0.77 KDM4E (0.38) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL30499285 0.77 BACE1 (0.57) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL11973788 0.77 BACE1 (0.57) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL2133059 0.76 NR4A2 (0.54) CYP1A2PDGFRBPDGFRA
SCHEMBL30506415 0.76 NR4A2 (0.54) CYP1A2PDGFRBPDGFRA
SCHEMBL5958458 0.76 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ACASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 163 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105037266-A Antibacterial chloroxoquinoline derivative WANG ZIHOU 2015-11-11 CN claimed
CN-105017145-A Chloroxoquinoline derivative with anti-tumor activity WANG ZIHOU 2015-11-04 CN claimed
CN-103864680-A Chloroxoquinoline derivative with antineoplastic activity WANG ZIHOU 2014-06-18 CN claimed
CN-103864681-A Chloroxoquinoline derivatives for antibacterial use WANG ZIHOU 2014-06-18 CN claimed
EP-0056765-B1 PREPARATION OF 4-HYDROXYQUINOLINES RHONE-POULENC SANTE (FR) 1985-06-19 EP claimed
EP-0056765-A1 Preparation of 4-hydroxyquinolines RHONE-POULENC SANTE (FR) 1982-07-28 EP claimed
CN-121426745-A Burisperidone Synthesis method of intermediate 鲁南制药集团股份有限公司 2026-01-30 CN disclosed
CN-119661537-A Nucleoside compound, preparation method thereof, composition thereof and application of nucleoside compound in medicine 中国科学院上海药物研究所 2025-03-21 CN disclosed
EP-3833668-B1 PRMT5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2025-03-19 EP disclosed
WO-2025044876-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND ORGANIC ELECTROLUMINESCENT ELEMENT COMPRISING SAME 海宁奕诺炜特科技有限公司 2025-03-06 WO disclosed
CN-114057815-B Novel 6-6 bicyclic aromatic ring substituted nucleosides as PRMT5 inhibitors 詹森药业有限公司 2025-02-25 CN disclosed
WO-2024238406-A1 FUROPYRIDINE COMPOUNDS AS P53 MUTANT STABILIZER AND USES THEREOF FRONTIER MEDICINES CORPORATION (US) 2024-11-21 WO disclosed
US-12145961-B2 Spirobicyclic analogues JANSSEN PHARMACEUTICA NV (BE) 2024-11-19 US disclosed
WO-2004014871-A1 VANILLOID RECEPTOR LIGANDS AND THEIR USE IN TREATMENTS AMGEN INC. (US) 2004-02-19 WO disclosed
EP-0097585-B1 PROCESS FOR THE PREPARATION OF 4-HYDROXY QUINOLINES RHONE-POULENC SANTE (FR) 1986-03-26 EP disclosed
EP-0056765-B1 PREPARATION OF 4-HYDROXYQUINOLINES RHONE-POULENC SANTE (FR) 1985-06-19 EP disclosed
EP-0056766-B1 PROCESS FOR THE PREPARATION OF 4-AMINO-CHLOROQUINOLINES RHONE-POULENC SANTE (FR) 1984-05-16 EP disclosed
EP-0097585-A1 Process for the preparation of 4-hydroxy quinolines RHONE-POULENC SANTE (FR) 1984-01-04 EP disclosed
EP-0056765-A1 Preparation of 4-hydroxyquinolines RHONE-POULENC SANTE (FR) 1982-07-28 EP disclosed
EP-0056766-A1 Process for the preparation of 4-amino-chloroquinolines RHONE-POULENC SANTE (FR) 1982-07-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12145961-B2 Spirobicyclic analogues PRMT5, HDAC5, SIRT5 ALDH1A1 1492/4885MEN1 849/4885KMT2A 251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.