SCHEMBL483970

SCHEMBL483970

Oc1ccc2nc(Cl)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.55
ESR1 P03372 6/20 0.55
TTR P02766 3/20 0.44
CYP1A2 P05177 1/20 0.43
ESRRB O95718 1/20 0.41
ESRRA P11474 1/20 0.41
HSD17B14 Q9BPX1 1/20 0.41
HSD17B10 Q99714 2/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
PFKFB3 Q16875 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7794275 0.98 ESR2 (0.53) ESR2ESR1TTRCYP1A2ESRRB
SCHEMBL622672 0.84 ALDH1A1 (0.50) ESR2ESR1TTRCYP1A2ESRRB
SCHEMBL4468871 0.78 PLAU (0.63) ESR2ESR1
SCHEMBL1060994 0.77 ESR2 (0.59) ESR2ESR1TTRCYP1A2HSD17B14
SCHEMBL29522954 0.77 ESR2 (0.59) ESR2ESR1TTRCYP1A2HSD17B14
SCHEMBL29447040 0.77 BACE1 (0.50) PDE3BPDE3AALDH1A1
SCHEMBL198060 0.77 BACE1 (0.50) PDE3BPDE3AALDH1A1
Bromide SCHEMBL23412828 0.77 PLAU (0.61) ESR2ESR1
SCHEMBL16500490 0.76 ESR1 (0.49) ESR2ESR1TTRCYP1A2HSD17B14
SCHEMBL27671114 0.76 ESR2 (0.57) ESR2ESR1TTRCYP1A2HSD17B14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 340 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119285543-B Sulfonylation method of halogenated quinoline and aryl sulfonyl hydrazine 南京工业大学 2026-05-15 CN claimed
CN-119285543-A Sulfonylation method of halogenated quinoline and aryl sulfonyl hydrazine 南京工业大学 2025-01-10 CN claimed
CN-103200820-B As the substd quinolines compound of GSNO reductase inhibitor Nivalis Therapeutics (US) 2016-04-06 CN claimed
CN-119285543-B Sulfonylation method of halogenated quinoline and aryl sulfonyl hydrazine 南京工业大学 2026-05-15 CN disclosed
US-20260125410-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS UNIV YALE (US) 2026-05-07 US disclosed
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS TORAY INDUSTRIES, INC. (JP) 2026-03-26 US disclosed
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof TORAY INDUSTRIES, INC. (JP) 2026-03-10 US disclosed
US-12528791-B2 Thyroid hormone receptor beta agonist compounds TERNS PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
US-20250388614-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS UNIV YALE (US) 2025-12-25 US disclosed
EP-4658263-A2 COMPOUNDS AND METHODS FOR TREATING, AMELIORATING, OR PREVENTING ARTHRITIS Yale University (US) 2025-12-10 EP disclosed
US-12485178-B2 Bifunctional small molecules to target the selective degradation of circulating proteins YALE UNIVERSITY (US) 2025-12-02 US disclosed
CN-1628109-A Novel aryl-and heteroaryl-piperazines NOVO NORDISK AS (DK) 2005-06-15 CN disclosed
WO-2005037285-A1 2,6-DISUBSTITUTED QUINAZOLINES, QUINOXALINES, QUINOLINES AND ISOQUINOLINES AS INHIBITORS OF RAF KINASE FOR TREATMENT OF CANCER CHIRON CORPORATION (US) 2005-04-28 WO disclosed
US-20050085482-A1 2,6-Disubstituted quinazolines, quinoxalines, quinolines and isoquinolines and methods of their use as inhibitors of RAF kinase CHIRON CORPORATION (US) 2005-04-21 US disclosed
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
EP-1474401-A2 NOVEL ARYL- AND HETEROARYLPIPERAZINES NOVO NORDISK A/S (DK) 2004-11-10 EP disclosed
US-20030236259-A1 Novel aryl- and heteroarylpiperazines HIGH POINT PHARMACEUTICALS, LLC 2003-12-25 US disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed
WO-2003066604-A2 NOVEL ARYL- AND HETEROARYLPIPERAZINES NOVO NORDISK A/S (DK) 2003-08-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085482-A1 2,6-Disubstituted quinazolines, quinoxalines, quinolines and isoquinolines and methods of their use as inhibitors of RAF kinase RAF1, BRAF, ARAF ESR2 3785/4885ESR1 4601/4885TTR 4864/4885
US-20030236259-A1 Novel aryl- and heteroarylpiperazines HRH3, HRH2, HRH4 ESR2 448/4885ESR1 703/4885TTR 4616/4885
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS AIFM2, GPX1, SOD1 ESR2 860/4885ESR1 3396/4885TTR 3107/4885
US-12485178-B2 Bifunctional small molecules to target the selective degradation of circulating proteins ASGR1, LDLR, FCGR2A ESR2 1540/4885ESR1 2058/4885TTR 257/4885
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof AIFM2, GPX1, GPX4 ESR2 411/4885ESR1 3178/4885TTR 4477/4885
US-12528791-B2 Thyroid hormone receptor beta agonist compounds THRB, THRA, TSHR ESR2 248/4885ESR1 1751/4885TTR 154/4885
US-20260125410-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS ASGR1, COL2A1, FCGR2A ESR2 219/4885ESR1 361/4885TTR 699/4885
US-20250388614-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS ASGR1, COL2A1, LDLR ESR2 335/4885ESR1 525/4885TTR 456/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.