SCHEMBL6229595

SCHEMBL6229595

CC(C)COC(=O)N1CCC(C(O)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.49
MAPT P10636 2/20 0.49
MAPK1 P28482 1/20 0.49
SLC6A3 Q01959 9/20 0.47
SLC6A2 P23975 7/20 0.47
SLC6A4 P31645 7/20 0.47
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
USP2 O75604 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 1/20 0.42
KIT P10721 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
TACR2 P21452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5705691 0.81 MAPT (0.52) HTTMAPTMAPK1SLC6A3ALDH1A1
SCHEMBL15794120 0.75 MAPT (0.44) HTTMAPTMAPK1SLC6A3SLC6A2
SCHEMBL1834064 0.74 RAB9A (0.48) ALDH1A1SMN1; SMN2TSHRKITL3MBTL1
SCHEMBL13503893 0.73 RAB9A (0.49) ALDH1A1SMN1; SMN2TSHRKITL3MBTL1
SCHEMBL5737424 0.72 HRH1 (0.60)
SCHEMBL1693088 0.71 RAB9A (0.44) MAPTALDH1A1SMN1; SMN2KITL3MBTL1
SCHEMBL3986658 0.70 HTT (0.41) HTTMAPTMAPK1SLC6A3SLC6A2
SCHEMBL4596054 0.70 GAA (0.45) MAPTALDH1A1LMNASMN1; SMN2L3MBTL1
SCHEMBL704010 0.70 RAB9A (0.51) ALDH1A1HPGDKITMEN1KMT2A
SCHEMBL4595299 0.69 RAB9A (0.41) HTTALDH1A1SMN1; SMN2KITL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517894-A1 N-BENZYL-3-PHENYL-3-HETEROCYCLYL-PROPIONAMIDE COMPOUNDS AS TACHYKININ ANTAGONISTS AND/OR SEROTONIN REUPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-03-30 EP disclosed
WO-2004005255-A1 N-BENZYL-3-PHENYL-3-HETEROCYCLYL-PROPIONAMIDE COMPOUNDS AS TACHYKININ AND/ OR SEROTONIN REUPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-01-15 WO disclosed