SCHEMBL6230832

SCHEMBL6230832

O=C(O)c1n[nH]c(-c2ccccc2F)c1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 3/20 0.44
CPB1 P15086 1/20 0.40
TSHR P16473 1/20 0.40
NPC1 O15118 2/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
BRD4 O60885 1/20 0.39
FFAR1 O14842 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715742 0.86 KDM4E (0.44) NPC1BRD4RAB9ASMN1; SMN2KDM4E
SCHEMBL6231126 0.81 IKBKE (0.42) PTGER1BRD4HTR1ASLC6A2SLC6A4
SCHEMBL4206891 0.77 NR4A2 (0.44) TSHRNR4A1NR4A2NR4A3KDM4E
SCHEMBL4205180 0.72 ALDH1A1 (0.55) TSHRNPC1RAB9ASMN1; SMN2NR4A1
SCHEMBL25037414 0.72 KDM4E (0.46) PTGER1NPC1MRGPRX4NR4A1NR4A2
SCHEMBL30038623 0.72 KDM4E (0.46) PTGER1NPC1MRGPRX4NR4A1NR4A2
SCHEMBL30862699 0.70 TSHR (0.45) PTGER1TSHRMRGPRX4KDM4EALDH1A1
SCHEMBL25037125 0.70 TSHR (0.45) PTGER1TSHRMRGPRX4KDM4EALDH1A1
SCHEMBL4224922 0.70 ALDH1A1 (0.53) TSHRNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL21312413 0.70 F10 (0.42) PTGER1CPB1TSHRFFAR1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003076443-A9 SPIRO COMPOUNDS WITH NPY ANTAGONISTIC ACTIVITY BANYU PHARMA CO LTD (JP) 2005-01-20 WO disclosed
EP-1483266-A1 SPIRO COMPOUNDS WITH NPY ANTAGONISTIC ACTIVITY BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-12-08 EP disclosed
WO-2003076443-A1 SPIRO COMPOUNDS WITH NPY ANTAGONISTIC ACTIVITY BANYU PHARMACEUTICAL CO., LTD. (JP) 2003-09-18 WO disclosed