SCHEMBL6231144

SCHEMBL6231144

CCN1CCCC1CN(CC1CCCCC1)c1nc(N)nc(Oc2ccc(N)cc2F)n1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ACHE P22303 1/20 0.30
HTR4 Q13639 1/20 0.30
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6429666 0.88 PIK3CD (0.34) ALDH1A1DRD2
SCHEMBL5550419 0.81 MAPT (0.33) KDM4EALDH1A1DRD2
SCHEMBL5549889 0.78 GALR1 (0.45) ALDH1A1
SCHEMBL4838866 0.77 DRD2 (0.40) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL6233417 0.77 GALR1 (0.38) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL6429807 0.74 HTT (0.39) KDM4EALDH1A1
SCHEMBL6612950 0.74 DRD2 (0.33) DRD2
SCHEMBL6233350 0.74
SCHEMBL5553491 0.73 GALR1 (0.46) DRD2
SCHEMBL6428940 0.73 PIK3CA (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560817-A1 METHODS AND COMPOSITIONS OF NOVEL TRIAZINE COMPOUNDS Reddy US Therapeutics, Inc. (US) 2005-08-10 EP claimed
WO-2004026844-A1 METHODS AND COMPOSITIONS OF NOVEL TRIAZINE COMPOUNDS REDDY US THERAPEUTICS, INC. (US) 2004-04-01 WO claimed
EP-1546134-A1 PIPERAZINE SUBSTITUTED ARYL BENZODIAZEPINES ELI LILLY AND COMPANY (US) 2005-06-29 EP disclosed
WO-2004014895-A1 PIPERAZINE SUBSTITUTED ARYL BENZODIAZEPINES ELI LILLY AND COMPANY (US) 2004-02-19 WO disclosed