SCHEMBL6232469

SCHEMBL6232469

COC1C(=O)NC(=O)N1C

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230625 0.75
SCHEMBL6233683 0.72 KDM4E (0.33)
SCHEMBL6232448 0.70 HSD11B1 (0.36)
SCHEMBL6232475 0.69 NPC1 (0.36)
SCHEMBL6235193 0.69 GAA (0.44)
SCHEMBL12570736 0.69
SCHEMBL20201458 0.69
SCHEMBL5956026 0.67
SCHEMBL5956305 0.67
SCHEMBL9775548 0.67 ADRA2C (0.33) ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0160618-A1 Hydantoin derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1985-11-06 EP claimed
JP-8134043-A None JP disclosed
EP-3639821-B1 CARCINOGENESIS INHIBITOR NAT CANCER CT (JP) 2024-08-28 EP disclosed
CN-110740729-B Carcinogenesis inhibitor 国立研究开发法人国立癌症研究中心 2023-05-16 CN disclosed
US-11464762-B2 Carcinogenesis inhibitor NATIONAL CANCER CENTER (JP) 2022-10-11 US disclosed
US-20200276163-A1 CARCINOGENESIS INHIBITOR NATIONAL CANCER CENTER (JP) 2020-09-03 US disclosed
EP-3639821-A1 CARCINOGENESIS INHIBITOR National Cancer Center (JP) 2020-04-22 EP disclosed
CN-110740729-A Carcinogenesis inhibitor 国立研究开发法人国立癌症研究中心 2020-01-31 CN disclosed
EP-1243261-B1 Use of a hydantoin derivative in a pharmaceutical composition against hypoalbuminaemia NIPPON ZOKI PHARMACEUTICAL CO (JP) 2005-04-27 EP disclosed
EP-1018339-B1 Use of hydantoin derivatives for the preparation of a medicament for the treatment of intractable vasculitis. NIPPON ZOKI PHARMACEUTICAL CO (JP) 2003-05-02 EP disclosed
US-6451831-B1 TREATMENT WITH HYDANTOIN DERIVATIVE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2002-09-17 US disclosed
US-6251929-B1 ADMINISTERING TO A PATIENT A HYDANTOIN DERIVATIVES AND SALTS AS THERAPEUTIC AND PREVENTIVE AGENTS FOR INTRACTABLE VASCULITIS SUCH AS MALIGNANT RHEUMATOID ARTHRITIS(MRA), PERIARTERITIS NODOSA, WEGENER'S GRANULOMATOSIS ETC. NIPPON ZOKI PHARMACEUTICALS CO., LTD. (JP) 2001-06-26 US disclosed
EP-0780125-B1 Use of hydantoin derivatives for the preparation of a medicament for the treatment of dieases associated with the presence of active oxygen and free radicals NIPPON ZOKI PHARMACEUTICAL CO (JP) 2001-04-18 EP disclosed
US-6197806-B1 USING A HYDANTOIN DERIVATIVE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2001-03-06 US disclosed
EP-1018339-A1 Therapeutic agent for intractable vasculitis NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2000-07-12 EP disclosed
EP-0780125-A2 Pharmaceutical composition containing a hydantoin derivative and use of said derivative NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-06-25 EP disclosed
JP-H08134043-A PRODUCTION OF 5-ALKOXYHYDANTOINS SUMITOMO SEIKA CHEM CO LTD 1996-05-28 JP disclosed
EP-0160618-B1 HYDANTOIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1991-08-14 EP disclosed
US-4647574-A Hypoglycemic hydantoin derivatives NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1987-03-03 US disclosed
EP-0160618-A1 Hydantoin derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1985-11-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11464762-B2 Carcinogenesis inhibitor APC, MKI67, HRAS ADRA2C 4868/4885
US-20200276163-A1 CARCINOGENESIS INHIBITOR APC, MKI67, HRAS ADRA2C 4868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.