SCHEMBL6232790

SCHEMBL6232790

Nc1ccnc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.50
NOS2 P35228 1/20 0.50
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
KMO O15229 1/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
XDH P47989 1/20 0.46
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
IDO1 P14902 1/20 0.44
IKBKB O14920 1/20 0.43
BRD4 O60885 1/20 0.43
SCN2A Q99250 1/20 0.43
CCNT1 O60563 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CDK9 P50750 1/20 0.43
MAPKAPK2 P49137 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19066984 0.85 NOS3 (0.50) NOS3NOS2ADORA2AADORA1KMO
SCHEMBL28946840 0.83 ADORA2A (0.51) ADORA2AADORA1NPC1RAB9AXDH
SCHEMBL7210508 0.81 IDO1 (0.53) KMONPC1RAB9AIDO1SCN2A
SCHEMBL2666275 0.81 KMO (0.48) KMONPC1RAB9AXDHIDO1
SCHEMBL29206336 0.81 KMO (0.48) ADORA2AADORA1KMONPC1RAB9A
SCHEMBL11390484 0.81 AURKA (0.47) ADORA2AADORA1KMONPC1RAB9A
SCHEMBL3794168 0.80 TRPV3 (0.48) NOS3NOS2
SCHEMBL13728192 0.79 KMO (0.52) KMO
SCHEMBL2885661 0.78 MEN1 (0.51) NPC1RAB9A
SCHEMBL28450652 0.78 KDM4E (0.56) ADORA2AADORA1KMONPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023242228-A1 4-SUBSTITUTED (1H-BENZO[D]IMIDAZOL-2-YL)-1H-PYRAZOLES AS BUB1 INHIBITORS USEFUL FOR TREATING CANCERS UNIVERSITEIT LEIDEN (NL) 2023-12-21 WO disclosed
EP-4112605-A1 PYRIMIDINE-2,4-DIAMINE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Anhui Medical University (CN) 2023-01-04 EP disclosed
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed