SCHEMBL6232942

SCHEMBL6232942

COC(=O)c1ccc2[nH]c(=O)c(-c3cccs3)nc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
LMNA P02545 1/20 0.58
GLA P06280 1/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
HSD17B10 Q99714 1/20 0.58
ERCC1 P07992 1/20 0.48
FEN1 P39748 1/20 0.48
ERCC4 Q92889 1/20 0.48
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
STK33 Q9BYT3 9/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
ATM Q13315 1/20 0.46
PARP1 P09874 1/20 0.44
RPS6KB2 Q9UBS0 2/20 0.44
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1905773 0.88 RAB9A (0.55) NPC1RAB9ALMNAGLACASP1
SCHEMBL5507978 0.86 NPC1 (0.64) NPC1RAB9ALMNAGLACASP1
SCHEMBL16390944 0.83 HSD17B10 (0.55) NPC1RAB9ALMNAGLACASP1
SCHEMBL6237123 0.82 ALDH1A1 (0.66) NPC1RAB9ALMNACASP1CASP7
SCHEMBL9960897 0.81 KDM4E (0.56) NPC1RAB9ALMNAALDH1A1HPGD
SCHEMBL1902589 0.81 CASP1 (0.64) NPC1RAB9ALMNAGLACASP1
SCHEMBL1903037 0.79 NPC1 (0.68) NPC1RAB9ALMNAGLACASP1
SCHEMBL1904092 0.79 NPC1 (0.58) NPC1RAB9ALMNAGLACASP1
SCHEMBL1905757 0.79 NPC1 (0.55) NPC1RAB9ALMNAGLACASP1
SCHEMBL1901859 0.77 NPC1 (0.68) NPC1RAB9ALMNAGLACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007099-A2 PKB INHIBITORS AS ANTI-TUMOR AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-27 WO disclosed