SCHEMBL6232949

SCHEMBL6232949

CN(CCCn1c(N(C)C)nc2cc(N)ccc21)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
RAD52 P43351 1/20 0.41
HTT P42858 1/20 0.41
BACE1 P56817 5/20 0.38
JAK2 O60674 2/20 0.37
JAK1 P23458 2/20 0.37
TYK2 P29597 2/20 0.37
JAK3 P52333 2/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
TLR8 Q9NR97 1/20 0.36
NUDT1 P36639 1/20 0.36
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NQO2 P16083 1/20 0.35
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6231516 0.93 KDM4E (0.43) KDM4ERAD52HTTBACE1JAK2
SCHEMBL6231518 0.85 KDM4E (0.43) KDM4ERAD52HTTBACE1JAK2
SCHEMBL6271695 0.83 KDM4E (0.41) KDM4ERAD52HTTHDAC1HDAC6
SCHEMBL6258152 0.72 KDM4E (0.40) KDM4ERAD52HTTBACE1HDAC6
SCHEMBL6604741 0.72 KDM4E (0.45) KDM4ERAD52HTTHDAC6TDP1
SCHEMBL6234983 0.70 KDM4E (0.45) KDM4ERAD52HTTTDP1TLR8
SCHEMBL17487511 0.70 CXCL8 (0.53) KDM4ERAD52HTTTDP1LMNA
SCHEMBL6233721 0.68 KDM4E (0.44) KDM4ERAD52HTTBACE1HDAC6
SCHEMBL18960395 0.68 NTRK1 (0.42) KDM4ERAD52HTT
SCHEMBL5226357 0.67 HDAC6 (0.48) KDM4EHTTHDAC1HDAC6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed