SCHEMBL6234983

SCHEMBL6234983

CN(C)c1nc2cc(N)ccc2n1C[CH]C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.45
RAD52 P43351 1/20 0.45
HTT P42858 2/20 0.41
ALDH1A1 P00352 5/20 0.35
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MEN1 O00255 1/20 0.33
CASP3 P42574 1/20 0.33
KMT2A Q03164 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CNR2 P34972 2/20 0.33
MAPT P10636 5/20 0.33
GFER P55789 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
HSD17B10 Q99714 2/20 0.32
NSD2 O96028 1/20 0.31
BRD4 O60885 1/20 0.31
NQO2 P16083 2/20 0.31
TLR8 Q9NR97 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271695 0.72 KDM4E (0.41) KDM4ERAD52HTTALDH1A1CNR2
SCHEMBL6604741 0.72 KDM4E (0.45) KDM4ERAD52HTTALDH1A1NPC1
SCHEMBL6231516 0.72 KDM4E (0.43) KDM4ERAD52HTTALDH1A1KMT2A
SCHEMBL6258152 0.71 KDM4E (0.40) KDM4ERAD52HTTALDH1A1KMT2A
SCHEMBL6232949 0.70 KDM4E (0.41) KDM4ERAD52HTTALDH1A1TDP1
SCHEMBL6231518 0.69 KDM4E (0.43) KDM4ERAD52HTTALDH1A1RAB9A
SCHEMBL18960395 0.69 NTRK1 (0.42) KDM4ERAD52HTTKMT2ACNR2
SCHEMBL17487511 0.69 CXCL8 (0.53) KDM4ERAD52HTTALDH1A1KMT2A
SCHEMBL623760 0.65 KDM4E (0.66) KDM4ERAD52HTTALDH1A1RAB9A
SCHEMBL6420487 0.65 KDM4E (0.50) KDM4ERAD52HTTALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed