SCHEMBL6233172

SCHEMBL6233172

CCOC(=O)CC1c2cc(C(C)(C)C)ccc2C(=O)N1CC(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.38
PIN4 Q9Y237 1/20 0.38
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MCL1 Q07820 1/20 0.36
IDO1 P14902 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
TNF P01375 1/20 0.34
DNMT1 P26358 3/20 0.33
LMNA P02545 2/20 0.33
BRD4 O60885 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27528495 0.91 CYP11B1 (0.43) PIN1PIN4IDO1CYP11B1CYP11B2
SCHEMBL6231541 0.87 PIN1 (0.41) PIN1PIN4IDO1CYP1A2LMNA
SCHEMBL4473163 0.85 MCL1 (0.39) CYP2C19MCL1TNFDNMT1ALDH1A1
SCHEMBL20000833 0.85 MCL1 (0.36) MCL1TNFDNMT1ALDH1A1HPGD
SCHEMBL6236384 0.85 ALDH1A1 (0.43) PIN1PIN4CYP11B1CYP11B2BRD4
SCHEMBL6234016 0.85 TDP2 (0.42) PIN1PIN4CYP2C9CYP2C19MCL1
SCHEMBL27528481 0.82 CYP11B1 (0.41) PIN1PIN4IDO1CYP11B1CYP11B2
SCHEMBL27528478 0.82 IDO1 (0.52) PIN1PIN4IDO1CYP1A2KDM4E
SCHEMBL13708551 0.81 MCL1 (0.34) MCL1TNFDNMT1ALDH1A1
SCHEMBL27552574 0.80 ALDH1A1 (0.44) PIN1PIN4CYP2C9CYP2C19IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1528923-A1 N-((3-OXO-2,3-DIHYDRO-1H-ISOINDOL-1-YL)ACETYL)GUANIDINE DERIVATIVES AS NHE1-INHIBITORS FOR THE TREATMENT OF INFARCTION AND ANGINA PECTORIS Aventis Pharma Deutschland GmbH (DE) 2005-05-11 EP disclosed
WO-2003101450-A1 N- ((3-OXO2, 3-DIHYDRO-1H-ISOINDOL-1-YL) ACETYL) GUANIDINE DERIVATIVES AS NHE-1 INHIBITORS FOR THE TREATMENT OF INFARCTION AND ANGINA PECTORIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-12-11 WO disclosed